2-Substituted 3-arylindoles through palladium-catalyzed arylative cyclization of 2-alkynyltrifluoroacetanilides with arylboronic acids under oxidative conditions.

نویسندگان

  • Antonio Arcadi
  • Sandro Cacchi
  • Giancarlo Fabrizi
  • Antonella Goggiamani
  • Antonia Iazzetti
  • Fabio Marinelli
چکیده

Free NH 2-substituted 3-arylindoles have been prepared usually in good to high yields through the palladium-catalyzed reaction of readily available 2-alkynyltrifluoroacetanilides with arylboronic acids under oxidative conditions. The reaction tolerates a variety of useful functional groups both in the arylboronic acid and in the alkyne, including chloro, formyl, and ester groups.

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منابع مشابه

Palladium-catalyzed cyclization of o-alkynyltrifluoroacetanilides followed by isocyanide insertion: synthesis of 2-substituted 1H-indole-3-carboxamides.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 11 4  شماره 

صفحات  -

تاریخ انتشار 2013